Home Neuronal Signaling -GPCR & G Protein -Transmembrane Transporters P2 Receptor P2Y receptor-Selectief Inhibitors | Antagonists | Modulators

P2Y receptor-Selectief Inhibitors | Antagonists | Modulators

  • P2X receptor
  • P2Y receptor
Cat.nr. Productnaam Informatie Selectief / Pan IC50 / Ki
S4079 Ticagrelor Ticagrelor is the first reversibly binding oral P2Y12 receptor antagonist with Ki of 2 nM. Selective P2Y12, Ki: 2 nM
S2855 MRS 2578 MRS2578 is a potent P2Y6 receptor antagonist with IC50 of 37 nM, exhibits insignificant activity at P2Y1, P2Y2, P2Y4,and P2Y11 receptors. Selective P2Y6, IC50: 37 nM
S1415 Clopidogrel Clopidogrel is an oral, thienopyridine class antiplatelet agent. Selective
S1258 Prasugrel Prasugrel is a thienopyridine ADP receptor (P2Y12) antagonist, used for the reduction of thrombotic cardiovascular events. Selective