Progesterone Receptor

기타 Endocrinology & Hormones 억제제

Adrenergic Receptor Androgen Receptor Estrogen/progestogen Receptor Aromatase 5-alpha Reductase RAAS Glucocorticoid Receptor ACE Mineralocorticoid Receptor PGDS

Cat.No.	제품명	정보	제품 사용 인용
S2567	Medroxyprogesterone Acetate (MPA)	MPA (Medroxyprogesterone acetate) is a synthetic progestin and act as a potent progesterone receptor agonist, used to treat abnormal menstruation or irregular vaginal bleeding.	Cancer Sci, 2025, 10.1111/cas.70081 Cell Prolif, 2024, e13780. J Transl Med, 2024, 22(1):478
S4040	Norethindrone	Norethindrone (Norethisterone) is a synthetic progestin, which mimic the actions of the endogenous ovarian hormone progesterone.	Nature Cancer, 2020, 235-248 Nat Cancer, 2020, 1(2):235-248
S2606	Mifepristone (RU-486)	Mifepristone is a remarkably active antagonist of progesterone receptor and glucocorticoid receptor with IC50 of 0.2 nM and 2.6 nM, respectively. Mifepristone promotes cell autophagy and apoptosis, decreases Bcl-2 level and increases Beclin1 level, accompanied by weakened interaction between Bcl-2 and Beclin1.Mifepristone (RU486) can be used to induce animal models of Spontaneous Abortion.	Alcoholism: Clinical and Experimental Research, May 2020, 1025-1036 Scientific Reports, March 24, 2020, 5363 Frontiers in Immunology, August 12, 2022, 863034
S1705	Progesterone	Progesterone is an endogenous steroid hormone involved in the menstrual cycle, pregnancy, and embryogenesis of humans and other species. This compound is a potent agonist of the nuclear progesterone receptor (nPR) with Kd of 1 nM; an agonist of the membrane progesterone receptors(mPRs); an antagonist of the σ1 receptor.	Bone Res, 2025, 13(1):37 Cell Proliferation, 2025, e70025 Nat Commun, 2024, 15(1):8708
S1304	Megestrol Acetate	Megestrol acetate (BDH1298, SC10363) is a synthetic progestogen, used to treat breast cancer and loss of appetite.	Scientific Reports, October 06, 2017, 12754 OncoTargets and Therapy, October 03, 2017, 4809-4819 iScience, 2024, 27(10):110862
S1251	Dienogest	Dienogest (STS 557) is an orally active synthetic progesterone, used for contraception and the treatment of endometriosis.	Texte Umweltbundesamt, June 2023, 81/2023 bioRxiv, July 13, 2023, nan Texte Umweltbundesamt, February 2026, 16/2026
S1377	Drospirenone	Drospirenone (ZK 3059) is a synthetic progestin that is an analog to spironolactone.	Acta Pharmaceutica Sinica B, 2023, 662-677 Acta Pharm Sin B, 2023, 13(2):662-677 Nature Cancer, 2020, 235-248
S3081	Ulipristal Acetate (CDB 2914)	Ulipristal acetate (CDB-2914, HRP 2000, RU 44675) is a selective SPRM for emergency contraception after an unprotected intercourse or contraceptive failure.	Nature, 2025, 10.1038/s41586-025-09684-7 The Journal of Clinical Endocrinology & Metabolism, 2019, 6256–6264 J Clin Endocrinol Metab, 2019, 104(12):6256-6264
S3635	Medroxyprogesterone	Medroxyprogesterone (MP) is a synthetic pregnane steroid and a derivative of progesterone. It is a potent progesterone receptor agonist.	Theranostics, 2024, 593-607
S3167	Altrenogest	Altrenogest (A35957, RU2267,R2267) is a progestogen structurally related to veterinary steroid trenbolone.
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