RSK2 Inhibitors

  • p70 S6K
  • p70 S6K1
  • RSK1
  • RSK2
  • RSK3
  • RSK4
Cat.No. 제품명 정보 선택적 / 팬 IC50 / Ki
S2843 BI-D1870 BI-D1870 is an ATP-competitive inhibitor of S6 ribosome for RSK1/2/3/4 with IC50 of 31 nM/24 nM/18 nM/15 nM, respectively; 10- to 100-fold selectivity for RSK than MST2, GSK-3β, MARK3, CK1 and Aurora B. Pan RSK2, IC50: 24 nM