| Cat.No. | 제품명 | 정보 | 선택적 / 팬 | IC50 / Ki |
|---|---|---|---|---|
| S2843 | BI-D1870 | BI-D1870 is an ATP-competitive inhibitor of S6 ribosome for RSK1/2/3/4 with IC50 of 31 nM/24 nM/18 nM/15 nM, respectively; 10- to 100-fold selectivity for RSK than MST2, GSK-3β, MARK3, CK1 and Aurora B. | Pan | RSK3, IC50: 18 nM |